Publications

40. Chatare, V. K., Andrade, R. B. Total Synthesis of (-)-Albocyclin, Angew. Chem. Int. Ed. 2017, 56, 5905 –5911

39. Zhao, S., Andrade, R. B. Development and Scope of the Arene-Fused Domino Michael/Mannich REaction: Application to the Total Syntheses of Aspidosperma Alkaloids (-)-Aspidospermidine, (-)-Tabersonine, (-)-Vincadifformine. JOC2017, 82, 521−531

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38. Zhao, S., Teijaro,C. N., Chen, H., Vaddypally, S. Zdilla, M., Andrade, R. B. Concise Syntheses of (-)-Sungucine, (-)-Isosungucine, and (-)-Strychnogucine B from (-)-Strychnine. Chem. Eur. J., 2016, 22, 11593–11596.

 

 

 

 

 

37. An, Y.; Doney, A. C.; Andrade, R. B.; Wheeler, S. E. Stacking Interactions between 9-Methyladenine and Heterocycles Commonly Found in Pharmaceuticals. J. Chem. Inf. Model, 2016, 56, 906-914.

36. Glassford, I., Teijaro, C. N., Daher, S. S., Weil, A., Redhu, S. K., Small, M. C., Buttaro, B., Nicholson, A. W., MacKerell, A. D. Jr., Cooperman, B. S., Andrade, R. B. Ribosome-templated azide-alkyne cycloadditions: synthesis of potent macrolide antibiotics by in situ click chemistry. JACS, 2016, 138, 3136-3144.

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35. Andrade, R. B. Total Synthesis of Desmethyl Macrolide Antibiotics. Synlett, 2015, 26, 2199-2215.

34. Kokkonda, P.; Brown, K. R.; Seguin, T. J.; Wheeler, S. E.; Vaddypally, S.; Zdilla, M. J.; Andrade, R. B. Biomimetic Total Syntheses of (−)-Leucoridines A and C through the Dimerization of (−)-Dihydrovalparicine. Angew. Chem. Int. Ed., 2015, 54, 12632-12635.

33. Teijaro, C. N.; Zhao, S.; Kokkonda, P.; Andrade, R. B. Total Syntheses of  (–)-Alstolucines A, B, and F, (–)-Echitamidine, and (–)-N-Demethylalstogucine. Synthesis 2015, 47, 1547–1556.

32. Teijaro, C. N.; Munagala, S.; Zhao, S.; Sirasani, G.; Kokkonda, P.; Malofeeva, E. V.; Hopper-Borge, E.; Andrade, R. B. Synthesis and Biological Evaluation of Pentacyclic Strychnos Alkaloids as Selective Modulators of the ABCC10 (MRP7) Efflux Pump. J. Med. Chem., 2014, 57, 10383–10390.

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31. Glassford, I.; Lee, M.; Wagh, B.; Velvadapu, V.; Paul, T.; Sandelin, G.; DeBrosse, C.; Klepacki, D.; Small, M.; C.; MacKerell, A. D., Jr.; Andrade, R. B. Desmethyl Macrolides: Synthesis and Evaluation of 4-Desmethyl Telithromycin. ACS Med. Chem. Lett., 2014, 5, 1021–1026.

30. Munagala, S.; Sirasani, G.; Kokkonda, P.; Phadke, M.; Krynetskaia, N.; Lu, P.; Sharom, F. J.; Chaudhury, S.; Abdulhameed, M. D. M.; Tawa, G.; Wallqvist, A.; Martinez, R.; Childers, W.; Abou-Gharbia, M.; Krynetskiy, E.; Andrade, R. B. Synthesis and evaluation of Strychnos alkaloids as MDR reversal agents for cancer cell eradication. Bioorg. Med. Chem., 2014, 22, 1148-1155.

29. Wagh, B.; Glassford, I.; Paul, T.; DeBrosse, C.; Klepacki, D.; Small, M.; C.; MacKerell, A. D., Jr.; Andrade, R. B. Desmethyl Macrolides: Synthesis and Evaluation of 4,8,10-Tridesmethyl Cethromycin. ACS Med. Chem. Lett., 2013, 4, 1114−1118.

28. Zhao, S.; Andrade, R. B. Domino Michael/Mannich/N-Alkylation Route to the Tetrahydrocarbazole Framework of Aspidosperma Alkaloids: Concise Total Syntheses of (−)-Aspidospermidine, (−)-Tabersonine, and (−)-Vincadifformine. J. Am. Chem. Soc. 2013, 135, 13334−13337

27. Sirasani, G.; Andrade, R. B. Total Synthesis of Strychnos Alkaloids Akuammicine, Strychnine, and Leuconicines A and B. In Strategies and Tactics in Organic Synthesis; Harmata, M., Ed. 2013, 9, 1−44.

26. Kaplan, J. M.; Shang, J.; Gobbo, P.; Antonello, S.; Armelao, L.; Chatare, V.; Ratner, D. M.; Andrade, R. B.; Maran, F. Confromationally Constrained Functional Peptide Monolayers for the Controlled Display of Bioactive Carbohydrate Ligands. Langmuir, 2013, 29, 8187-8192.

25. Zhao, S.; Sirasani, G.; Vaddypally, S.; Zdilla, M.; Andrade, R. B. Total Synthesis of (-)-Melotenine A. Angew. Chem. Int. Ed. 2013, 52, 8309−8311.

24. Small, M. C.; Lopes, P.; Andrade, R. B.; MacKerell, A. D., Jr. Impact of ribosomal modification on the binding of the antibiotic telithromycin using a combined Grand Canonical Monte Carlo/Molecular Dynamics simulation approach. PLoS Comput. Biol. 2013, 9, e1003113.

23. Wagh, B.; Glassford, I.; Paul, T.; DeBrosse, C.; Klepacki, D.; Small, M.; C.; MacKerell, A. D., Jr.; Andrade, R. B. Desmethyl Macrolides: Synthesis and Evaluation of 4,8-Didesmethyl Telithromycin. ACS Med. Chem. Lett., 2012, 3, 1013−1018.

22. Yu, A.; Shang, J.; Cheng, F.; Paik, B. A.; Kaplan, J. M.; Andrade, R. B.; Ratner, D. M. Biofunctional Paper via the Covalent Modification of Cellulose. Langmuir, 2012, 28, 11265–11273.

21. Velvadapu, V.; Glassford, I.; Lee, M.; Paul, T.; DeBrosse, C.; Klepacki, D.; Small, M.; C.; MacKerell, A. D., Jr.; Andrade, R. B. Desmethyl Macrolides: Synthesis and Evaluation of 4,10-Didesmethyl Telithromycin. ACS Med. Chem. Lett., 2012, 3, 211-215.

20. Shang, J.; Cheng, F.; Dubey, M.; Kaplan, J.; Rawal, M.; Jiang, X.; Newburg, D.; Sullivan, P. A.; Andrade, R. B.; Ratner, D. M. An organophosphonate strategy for functionalizing silicon photonic biosensors. Langmuir 2012, 28, 3338-3344.

19. Velvadapu, V.; Paul, T.; Wagh, B.; Glassford, I.; DeBrosse, C.; Andrade, R. B. Total Synthesis of (-)-4,8,10-Tridesmethyl Telithromycin. J. Org. Chem. 2011, 76, 7516-7527.

18. Sirasani, G.; Andrade, R. B. Total Synthesis of (-)-Leuconicine A and B. Org. Lett. 2011, 13, 4736-4737.

17. Sirasani, G.; Paul, T.; Andrade, R. B. Sequencing cross-metathesis and non-metathesis reactions to rapidly access building blocks for synthesis. Tetrahedron 2011, 67, 2197-2205.

16. Velvadapu, V.; Paul, T.; Wagh, B.; Klepacki, D.; Guvench, O.; MacKerell, A. Jr.; Andrade, R. B. Desmethyl Macrolides: Synthesis and Evaluation of 4,8,10-Tridesmethyl Telithromycin. ACS Med. Chem. Lett. 2011, 2, 68-72.

15. Sirasani, G.; Paul, T.; Dougherty, W., Jr.; Kassel, S.; Andrade, R. B. Concise Total Syntheses of (+/-)-Strychnine and (+/-)-Akuammicine. J. Org. Chem. 2010, 75, 3529–3532.

14. Sirasani, G.; Paul, T.; Andrade, R. B. Total Synthesis of (+)-Crocacin C. Bioorg. Med. Chem. 2010, 18, 3648-3655.

13. Andrade, R. B. Syntheses of the Crocacins. A Review. Org. Prep. Proced. Int. 2009, 41, 359-383.

12. Fortin, M.; Pham, K.; Kaplan, J.; Kirk, S.; Andrade, R. B. Gem-Dimethyl 4-Pentenyl Glycosides: Novel Glycosylating Agents and Anomeric Protecting Groups. Org. Lett. 2009, 11, 3594–3597.

11. Sirasani, G.; Andrade, R. B. Sequential One-Pot Cyclizations: Concise Access to the ABCE Tetracyclic Framework of Strychnos Alkaloids. Org. Lett. 2009, 11, 2085-2088.

10. Sirasani, G.; Paul, T.; Andrade, R. B. Concise asymmetric synthesis of (+)-Crocacin C. J. Org. Chem. 2008, 73, 6386-6388.

9. Paul, T.; Sirasani, G.; Andrade, R. B. One-pot sequential cross-metathesis/hydride reduction: highly stereoselective synthesis of primary (E)-allylic alcohols from terminal olefins. Tetrahedron Lett. 2008, 49, 3363-3367.

8. Andrade, R. B. Key Strategies in Glycan Synthesis Wiley Encyclopedia of Chemical Biology. 2008.

7. Velvadapu, V.; Andrade, R. B. Concise Syntheses of D-Desosamine, 2-Thiopyrimidinyl Desosamine Donors and Methyl Desosaminide Analogues from D-Glucose. Carb. Res., 2008, 343, 145–150.

6. Paul, T.; Andrade, R. B. Sequential cross-metathesis/phosphorus-based olefination: stereoselective synthesis of 2,4-dienoates. Tetrahedron Lett. 2007, 48, 5367-5370.

5. Andrade, R. B.; Martin, S. F. Formal Syntheses of (±)-Pinnaic Acid and (±)-Halichlorine. Org. Lett. 2005, 7, 5733-5735.

4. Love, K. R.; Andrade, R. B.; Seeberger, P. H. Linear Synthesis of a Protected H-Type II Pentasaccharide Using Glycosyl Phosphate Building Blocks. J. Org. Chem. 2001, 66, 8165-8176.

3. Plante, O. J.; Palmacci, E. R.; Andrade, R. B.; Seeberger, P. H. Oligosaccharide Synthesis with Glycosyl Phosphate and Dithiophosphate Triesters as Glycosylating Agents. J. Am. Chem. Soc. 2001, 123, 9545-9554.

2. Andrade, R. B.; Plante, O. J.; Melean, L. G.; Seeberger, P. H. Solid-Phase Oligosaccharide Synthesis: Preparation of Complex Structures Using a Novel Linker and Different Glycosylating Agents. Org. Lett. 1999, 1, 1811-1814.

1. Plante, O. J.; Andrade, R. B.; Seeberger, P. H. Synthesis and Use of Glycosyl Phosphates as Glycosyl Donors. Org. Lett. 1999, 1, 211-214.

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